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Synthesis of axially chiral biaryl thioglycosides through thiosugar-directed Pd-catalyzed asymmetric C–H activation
Franck Le Bideau
,
Maha Fatthalla
,
Nicolas Grimblat
,
Etienne Brachet
,
Mouad Alami
et al.
Journal articles
hal-03386143v1
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Visible light C-H amidation of heteroarenes with benzoyl azides
Etienne Brachet
,
T. Ghosh
,
I. Ghosh
,
B König
Journal articles
hal-02418685v1
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Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist
Etienne Brachet
,
Philippe Belmont
Journal articles
hal-02384634v1
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Nickel-Catalyzed Arylation, Alkenylation, and Alkynylation of Unprotected Thioglycosides at Room Temperature
Etienne Brachet
,
Jean-Daniel Brion
,
Mouad Alami
,
Samir Messaoudi
Journal articles
istex
hal-03073844v1
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Pd-Catalyzed Reaction of Sterically Hindered Hydrazones with Aryl Halides: Synthesis of Tetra-Substituted Olefins Related to iso -Combretastatin A4
Etienne Brachet
,
Abdallah Hamze
,
Jean-François Peyrat
,
Jean-Daniel Brion
,
Mouad Alami
et al.
Journal articles
hal-03073857v1
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Neuropilin 1 and Neuropilin 2 gene invalidation or pharmacological inhibition reveals their relevance for the treatment of metastatic renal cell carcinoma
Aurore Dumond
,
Etienne Brachet
,
Jérôme Durivault
,
Valérie Vial
,
Anna Puszko
et al.
Journal articles
hal-03132345v1
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A palladium-catalyzed coupling of 3-chloroquinoxalinones with various nitrogen-containing nucleophiles
Etienne Brachet
,
Jean-François Peyrat
,
Jean-Daniel Brion
,
Samir Messaoudi
,
Mouâd Alami
et al.
Journal articles
hal-03073852v1
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Synthesis, biological evaluation, and structure–activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors
Jessy Aziz
,
Etienne Brachet
,
Abdallah Hamze
,
Jean-François Peyrat
,
Guillaume Bernadat
et al.
Journal articles
hal-03073854v1
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Synthesis of axially chiral biaryl thioglycosides through thiosugar-directed Pd-catalyzed asymmetric C–H activation
Maha Fatthalla
,
Nicolas Grimblat
,
Etienne Brachet
,
Mouad Alami
,
Vincent Gandon
et al.
Journal articles
hal-03425421v1
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Light on Unsaturated Hydrocarbons - “Gotta Heterofunctionalize Them All”
Doriane Menigaux
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-03073829v1
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Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist
Etienne Brachet
,
Philippe Belmont
Journal articles
hal-03073838v1
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Visible light amination/Smiles cascade: access to phthalazine derivatives
Etienne Brachet
,
Leyre Marzo
,
Mohamed Selkti
,
Burkhard König
,
Philippe Belmont
et al.
Journal articles
hal-02384218v1
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Silver-catalyzed tandem cycloisomerization/hydroarylation reactions and mechanistic investigations for an efficient access to 1,2-dihydroisoquinolines
Maxime de Abreu
,
Yue Tang
,
Etienne Brachet
,
Mohamed Selkti
,
Véronique Michelet
et al.
Journal articles
hal-03132346v1
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Stereoselective Palladium-Catalyzed Alkenylation and Alkynylation of Thioglycosides
Etienne Brachet
,
Jean-Daniel Brion
,
Mouad Alami
,
Samir Messaoudi
Journal articles
istex
hal-03073842v1
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Palladium-Catalyzed Cross-Coupling of 1-Aminoazoles with Aryl Chlorides: Application to the Synthesis of Unsymmetrical N,N′ -Diaryl-1-aminoindoles
Etienne Brachet
,
Samir Messaoudi
,
Jean-François Peyrat
,
Jean-Daniel Brion
,
Mouad Alami
et al.
Journal articles
istex
hal-03073855v1
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Synthesis, 3D-structure and stability analyses of NRPa-308, a new promising anti-cancer agent
Etienne Brachet
,
Aurore Dumond
,
Wang-Qing Liu
,
Marie Fabre
,
Mohamed Selkti
et al.
Journal articles
hal-02418648v1
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Palladium-Catalyzed Coupling of N -Aminoazoles with 3-Halo-Substituted Quinolin-2(1 H )-ones, Coumarins, Quinoxalin-2(1 H )-ones, and Chromenes
Thi Thanh Huyen Luong
,
Etienne Brachet
,
Jean-Daniel Brion
,
Samir Messaoudi
,
Mouâd Alami
et al.
Journal articles
istex
hal-03073839v1
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Palladium-Catalyzed Cross-Coupling Reaction of Thioglycosides with (Hetero)aryl Halides
Etienne Brachet
,
Jean-Daniel Brion
,
Samir Messaoudi
,
Mouad Alami
Journal articles
istex
hal-03073850v1
|
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Spotlight on Photo‐Induced Aryl Migration Reactions.
Marie Huynh
,
Maxime de Abreu
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-03073199v1
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Synergistic Photoredox/Transition-Metal Catalysis for Carbon-Carbon Bond Formation Reactions
Maxime de Abreu
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-02384360v1
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Synergistic Photoredox/Transition-Metal Catalysis for Carbon-Carbon Bond Formation Reactions
Maxime de Abreu
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-03073824v1
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Visible light amination/Smiles cascade: access to phthalazine derivatives
Etienne Brachet
,
Leyre Marzo
,
Mohamed Selkti
,
Burkhard König
,
Philippe Belmont
et al.
Journal articles
hal-03073836v1
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Light-Enabled Radical 1,4-Aryl Migration Via a Phospho-Smiles Rearrangement
Maxime de Abreu
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-03132343v1
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Phosphine-Triggered Selectivity Switch in Silver-Catalyzed o -Alkynylbenzohydroxamic Acid Cycloisomerizations
Xavier Bantreil
,
Aurélie Bourderioux
,
Pierre Mateo
,
Caroline Hagerman
,
Mohamed Selkti
et al.
Journal articles
hal-03534140v1
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Phosphoramidates as Transient Precursors of Nitrogen‐Centered Radical Under Visible‐Light Irradiation: Application to the Synthesis of Phthalazine Derivatives
Maxime de Abreu
,
Mohamed Selkti
,
Philippe Belmont
,
Etienne Brachet
Journal articles
hal-03073822v1
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Visible Light-Induced Regioselective Cycloaddition of Benzoyl Azides and Alkenes To Yield Oxazolines
Peter Bellotti
,
Julien Brocus
,
Fatima El Orf
,
Mohamed Selkti
,
Burkhard König
et al.
Journal articles
hal-02384322v1
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